GPCR agonist-2 [291528-35-3]
Référence T60074-1ml
Conditionnement : 1mLx10mM(inDMSO)
Marque : TargetMol
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GPCR agonist-2
(Synonyms: 4-(Cyclopropylamino)-3-nitrobenzoic acid) Copy Product Info
GPCR agonist-2 (4-(Cyclopropylamino)-3-nitrobenzoic acid) is an agonist of the orphan human GPCR GPR109B.
Cas No. 291528-35-3
For research use only—not for human use. No sales to individuals. Use as intended only.
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Purity:99.96%
Appearance:Solid
Color:Yellow
COA HNMR LCMS
Product Introduction
GPCR agonist-2 AI Summary
GPCR agonist-2 exhibits agonist activity at the human GPR109b receptor when transfected in CHOK1 cells. Its bioactivity is demonstrated by the reversal of forskolin-induced cAMP elevation in a whole cell assay, with an EC50 value of 309.03 nM..
Note: Summary generated by AI. Data source: ChEMBL 
Bioactivity
Chemical Properties
Storage & Solubility Information
| Description | GPCR agonist-2 (4-(Cyclopropylamino)-3-nitrobenzoic acid) is an agonist of the orphan human GPCR GPR109B. |
| Synonyms | 4-(Cyclopropylamino)-3-nitrobenzoic acid |
| Molecular Weight | 222.2 |
| Formula | C10H10N2O4 |
| Cas No. | 291528-35-3 |
| Smiles | N(=O)(=O)C1=C(NC2CC2)C=CC(C(O)=O)=C1 |
| Storage | Powder: -20°C for 3 years | In solvent: -80°C for 1 year Shipping with blue ice/Shipping at ambient temperature. | |||||||||||||||||||||||||||||||||||
| Solubility Information | DMSO: 50 mg/mL (225.02 mM), Sonication is recommended.  | |||||||||||||||||||||||||||||||||||
Solution Preparation Table | ||||||||||||||||||||||||||||||||||||
DMSO
Note : The dilution table applies only to solid products. For liquid products, please calculate the stock solution based on the stated concentration and/or density. | ||||||||||||||||||||||||||||||||||||