PG 106 acetate
Référence TP1952L-10mg
Conditionnement : 10mg
Marque : TargetMol
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PG 106 acetate
(Synonyms: PG 106 acetate(944111-22-2 Free base)) Copy Product Info
PG 106 acetate is an effective and selective antagonist of the human melanocortin 3 (hMC3) receptor with an IC50 of 210 nM. PG 106 acetate has no activity with the hMC5 receptor and hMC4 receptors with an EC50 of 9900 nM.
For research use only—not for human use. No sales to individuals. Use as intended only.
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Purity:99.93%
Appearance:Solid
Color:White
COA LCMS MS
Product Introduction
Bioactivity
Chemical Properties
Storage & Solubility Information
| Description | PG 106 acetate is an effective and selective antagonist of the human melanocortin 3 (hMC3) receptor with an IC50 of 210 nM. PG 106 acetate has no activity with the hMC5 receptor and hMC4 receptors with an EC50 of 9900 nM. |
| Targets & IC50 | MC3R (human):210 nM |
| Synonyms | PG 106 acetate(944111-22-2 Free base) |
| Molecular Weight | 1068.23 |
| Formula | C53H73N13O11 |
| Smiles | CCCCC(NC(C)=O)C(N[C@H]1CC(NCCCC[C@@H](C(N)=O)NC([C@H](CC2=CNC3=CC=CC=C32)NC([C@H](CCC/N=C(N)\N)NC([C@@H](CC4=CC5=CC=CC=C5C=C4)NC(CCNC1=O)=O)=O)=O)=O)=O)=O.CC(O)=O |
| Sequence | Ac-Nle-Asp-Bal-{DL-2Nal}-{DL-Arg}-Trp-Lys (Bridge:Asp3-Lys8) |
| Sequence Short | XDXXRWK |
| Storage | Keep away from moisture Powder: -20°C for 3 years | In solvent: -80°C for 1 year Shipping with blue ice/Shipping at ambient temperature. |